Elagolix sodium

CAS No. 832720-36-2

Elagolix sodium ( NBI-56418 sodium )

Catalog No. M20990 CAS No. 832720-36-2

Elagolix sodium is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM respectively).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 34 In Stock
5MG 55 In Stock
10MG 87 In Stock
25MG 158 In Stock
50MG 258 In Stock
100MG 402 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Elagolix sodium
  • Note
    Research use only not for human use.
  • Brief Description
    Elagolix sodium is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM respectively).
  • Description
    Elagolix sodium is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM respectively).
  • Synonyms
    NBI-56418 sodium
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    GNRHR
  • Research Area
    Cancer
  • Indication
    Uterine leiomyoma

Chemical Information

  • CAS Number
    832720-36-2
  • Formula Weight
    653.57
  • Molecular Formula
    C32H29F5N3NaO5
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:50 mg/mL (76.50 mM); H2O:50 mg/mL (76.50 mM)
  • SMILES
    COc1cccc(-c2c(C)n(Cc3c(F)cccc3C(F)(F)F)c(=O)n(CC(NCCCC(=O)[O-])c3ccccc3)c2=O)c1F.[Na+]
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Barra F Scala C Ferrero S2.Elagolix sodium for the treatment of women with moderate to severe endometriosis-associated pain.Drugs Today (Barc). 2019 Apr;55(4):237-246.
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